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Palmitoylethanolamide: A Multifunctional Molecule for Neuroprotection, Chronic Pain, and Immune Modulation

Valeria Di Stefano, Luca Steardo Jr, Martina D'Angelo, Francesco Monaco, Luca Steardo. Biomedicines. 2025 May 22;13(6):1271.

ReviewHumansOther animals

Design
Review
Subjects
Not applicable; this is a narrative review, not a single study
Dose used in the study
Not applicable; this is a narrative review, not a single study
Duration
Not applicable; this is a narrative review, not a single study
What was measured
How palmitoylethanolamide and ultramicronised PEA (umPEA) are thought to work, and what the evidence shows for neuroprotection, chronic pain and immune modulation

What the authors reported

The review describes PEA acting mainly through PPAR-alpha, with additional effects via CB1/CB2, GPR55 and TRPV1. Ultramicronised PEA has improved bioavailability, and in the preclinical and clinical studies cited it reduces neuroinflammation, stabilises mast cells and enhances endocannabinoid system activity, with what the authors describe as a well-established safety profile.

Limits of this study

A narrative review summarising other studies, not new data of its own; it does not independently verify the claims it summarises. The authors declare no conflicts of interest.

Source

PubMed 40563990 · doi:10.3390/biomedicines13061271

Entry checked against the abstract on PubMed on 2026-09-22. The dose shown is the dose the researchers used. It is not a recommendation. How to read this page.